Arzoxifene (LY353381) is an orally active selective estrogen receptor modulator (SERM) with a fixed ring structure similar to raloxifene. It exhibits potent antiestrogenic effects on breast cancer and endometrium with minimal side effects and provides beneficial estrogenic effects on bone health and lipid profile.
Molekulargewicht:
475.6
CAS Nummer:
[182133-25-1]
Formel:
C28H29NO4S
Target-Kategorie:
Others|||Estrogen Receptor/ERR
T39259
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