(R)-GSK-3685032 is the R-enantiomer of GSK-3685032, a first-in-class, non-time-dependent, non-covalent, reversible, selective DNMT1 inhibitor with an IC50 of 0.036 µM, which induces robust loss of DNA methylation, transcriptional activation, and inhibition of cancer cell growth.
Molekulargewicht:
420.54
CAS Nummer:
[2170140-50-6]
Formel:
C22H24N6OS
Target-Kategorie:
Others|||DNA Methyltransferase
T39648
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