Emedastine, CAS [[87233-61-2]]

Produktübersicht

• Artikelname: Emedastine, CAS [[87233-61-2]]
• Artikelnummer: TGM-T3979
• Hersteller Artikelnummer: T3979
• Alternativnummer: TGM-T3979-1MLX10MM(INDMSO),TGM-T3979-1MG,TGM-T3979-5MG,TGM-T3979-10MG,TGM-T3979-25MG,TGM-T3979-50MG,TGM-T3979-100MG,TGM-T3979-500MG
• Hersteller: TargetMol
• Kategorie: Biochemikalien
• Alternative Synonym: LY188695 , Emadine

Produktbeschreibung

Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity. Emedastine reversibly and competitively blocks histamine by binding to H1 receptors, thus blocking its downstream activity. As a result this agent interferes with mediator release from mast cells either by inhibiting calcium ion influx across mast cell/basophil plasma membrane or by inhibiting intracellular calcium ion release within the cells. In addition, emedastine may also inhibit the late-phase allergic reaction mediated through leukotrienes or prostaglandins, or by producing an anti-platelet activating factor effect. Upon ocular administration, emedastine causes a dose-dependent inhibition of histamine-stimulated vascular permeability in the conjunctiva. Emedastine does not affect adrenergic, dopamine, or serotonin receptors.

Produkteigenschaften

• Molekulargewicht: 302.41
• Reinheit: 95.03%
• CAS Nummer: [87233-61-2]
• Formel: C17H26N4O
• Target-Kategorie: Histamine Receptor

Bilder

T3979