CDK7-IN-6 is a highly effective and specific inhibitor (IC50 100 nM) of cyclin-dependent kinase 7 (CDK7). It showcases remarkable selectivity, with more than a 200-fold preference for CDK7 over CDK1, CDK2, and CDK5. This compound holds significant potential for cancer research purposes.
Molekulargewicht:
524.07
CAS Nummer:
[2378710-04-2]
Formel:
C26H34ClN9O
Target-Kategorie:
Others|||CDK
T39943
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