MS67 is a potent and selective degrader of WD40 repeat domain protein 5 (WDR5) with a dissociation constant (Kd) of 63 nM, exhibiting no activity against protein methyltransferases, kinases, G-protein-coupled receptors (GPCRs), ion channels, and transporters, and notably demonstrating significant anticancer properties.
Molekulargewicht:
1030.14
CAS Nummer:
[2407452-77-9]
Formel:
C52H59F4N9O7S
Target-Kategorie:
PROTACs|||Histone Methyltransferase
T39976
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