Lesogaberan napadisylate, CAS [[477956-38-0]]

Produktübersicht

• Artikelname: Lesogaberan napadisylate, CAS [[477956-38-0]]
• Artikelnummer: TGM-T40572
• Hersteller Artikelnummer: T40572
• Alternativnummer: TGM-T40572-5MG
• Hersteller: TargetMol
• Kategorie: Biochemikalien
• Alternative Synonym: AZD-3355 napadisylate

Produktbeschreibung

Lesogaberan (AZD-3355) napadisylate is a potent and selective agonist of GABA B receptors, with an EC50 of 8.6 nM for human recombinant GABA B receptors. It has an affinity (Ki) of 5.1 nM for rat GABA B receptors and 1.4 µM for GABA A receptors, determined by displacement of [3H]GABA binding in brain membranes. Lesogaberan napadisylate exerts a peripheral mode of action, inhibiting transient lower esophageal sphincter relaxation.

Produkteigenschaften

• Molekulargewicht: 349.31
• CAS Nummer: [477956-38-0]
• Formel: C13H17FNO5PS
• Target-Kategorie: Others|||GABA Receptor

Bilder

T40572