Sulfaphenazole, CAS [[526-08-9]]

Produktübersicht

• Artikelname: Sulfaphenazole, CAS [[526-08-9]]
• Artikelnummer: TGM-T4567
• Hersteller Artikelnummer: T4567
• Alternativnummer: TGM-T4567-1MLX10MM(INDMSO),TGM-T4567-100MG
• Hersteller: TargetMol
• Kategorie: Biochemikalien
• Alternative Synonym: Plisulfan , Raziosulfa , Depocid , Depotsulfonamide

Produktbeschreibung

Sulfaphenazole (Plisulfan) is an inhibitor of CYP2C9 (Ki: 0.3 µM) that demonstrates at least 100-fold selectivity over other CYP450 isoforms (Ki: 63/29 µM for CYP2C8/CYP2C18, respectively, and no activity at CYP1A1, CYP1A2, CYP3A4, CYP2C19). At 10 µM, sulfaphenazole has been shown to inhibit endothelium-derived hyperpolarizing factor synthase, a CYP450 isozyme in the porcine coronary artery homologous to CYP2C8/9 that generates reactive oxygen species in coronary endothelial cells and modulates vascular tone and homeostasis.

Produkteigenschaften

• Molekulargewicht: 314.36
• Reinheit: 0.9997
• CAS Nummer: [526-08-9]
• Formel: C15H14N4O2S
• Target-Kategorie: Cytochromes P450|||Apoptosis|||Necroptosis|||Antibacterial|||Antibiotic

Bilder

T4567