CP681301 is a potent inhibitor of CDK5 with antiproliferative activity. CP681301 exhibits anti-tumor activity in Drosophila. CP681301 decreases the expression of CD133, OLIG2, SOX2, KI67, pCDK5 protein level in Glioma stem cells (GSCs). CP681301 reduces self-renewal in mouse glioma xenografts [1].
Molekulargewicht:
298.38
CAS Nummer:
[865317-32-4]
Formel:
C17H22N4O
Target-Kategorie:
Others|||DNA/RNA Synthesis|||CDK
T60661
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