Fasudil dihydrochloride, CAS [[203911-27-7]]

Artikelnummer: TGM-T61382
Artikelname: Fasudil dihydrochloride, CAS [[203911-27-7]]
Artikelnummer: TGM-T61382
Hersteller Artikelnummer: T61382
Alternativnummer: TGM-T61382-10MG,TGM-T61382-25MG,TGM-T61382-50MG,TGM-T61382-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
Alternative Synonym: HA1077 dihydrochloride , AT-877 dihydrochloride , AT877 dihydrochloride , HA-1077 dihydrochloride
Fasudil dihydrochloride, also known as HA-1077 and AT877, is a nonspecific inhibitor of RhoA/ROCK. Fasudil dihydrochloride exhibits inhibitory effects on protein kinases including ROCK1 (Ki = 0.33 µM), ROCK2 (IC50 = 0.158 µM), PKA (IC50 = 4.58 µM), PKC (IC50 = 12.30 µM), and PKG (IC50 = 1.650 µM), while also acting as a potent Ca2+ channel blocker and vasodilator, providing a multifunctional pharmacological tool for vascular, cardiovascular, and cellular signaling research.
Molekulargewicht: 364.29
Reinheit: 99.86%
CAS Nummer: [203911-27-7]
Formel: C14H19Cl2N3O2S
Target-Kategorie: ROCK|||Rho|||PKA|||PKC
T61382
T61382