CXCR4 antagonist 5, CAS [[2304749-86-6]]

Produktübersicht

• Artikelname: CXCR4 antagonist 5, CAS [[2304749-86-6]]
• Artikelnummer: TGM-T61419
• Hersteller Artikelnummer: T61419
• Alternativnummer: TGM-T61419-25MG,TGM-T61419-50MG,TGM-T61419-100MG
• Hersteller: TargetMol
• Kategorie: Biochemikalien

Produktbeschreibung

CXCR4 antagonist 5 (compound 23), a potent CXCR4 antagonist, exhibits high inhibition efficacy against CXCR4 with an IC50 value of 8.8 nM. It effectively suppresses CXCL12-induced cytosolic calcium increase (IC50 = 0.02 nM) and hinders CXCR4/CXCL12-mediated chemotaxis. Moreover, Compound 23 demonstrates favorable physicochemical properties and in vitro safety profiles, exhibiting only marginal to moderate inhibition of CYP isozymes and hERG [1].

Produkteigenschaften

• Molekulargewicht: 366.5
• CAS Nummer: [2304749-86-6]
• Formel: C21H30N6
• Target-Kategorie: Others|||CXCR

Bilder

T61419