GSK2646264, CAS [[1398695-47-0]]

Artikelnummer: TGM-T61527
Artikelname: GSK2646264, CAS [[1398695-47-0]]
Artikelnummer: TGM-T61527
Hersteller Artikelnummer: T61527
Alternativnummer: TGM-T61527-25MG,TGM-T61527-50MG
Hersteller: TargetMol
Kategorie: Biochemikalien
GSK2646264 (Compound 44) is a highly effective and specific inhibitor of spleen tyrosine kinase (SYK) with a pIC50 of 7.1. It also inhibits multiple kinases, including LCK (pIC50 5.4), LRRK2 (pIC50 5.4), GSK3beta (pIC50 5.3), JAK2 (pIC50 5), VEGFR2 (pIC50 4.5), Aurora B (pIC50 <4.6), and Aurora A (pIC50 <4.3). Notably, GSK2646264 demonstrates skin penetrability, reaching both the epidermis and dermis [1].
Molekulargewicht: 374.48
CAS Nummer: [1398695-47-0]
Formel: C24H26N2O2
Target-Kategorie: Others|||LRRK2|||JAK|||VEGFR|||Aurora Kinase|||GSK-3|||Syk|||Src
T61527