GABAA receptor agent 5, CAS [[1808389-92-5]]
Artikelnummer:
TGM-T61668
| Artikelname: |
GABAA receptor agent 5, CAS [[1808389-92-5]] |
| Artikelnummer: |
TGM-T61668 |
| Hersteller Artikelnummer: |
T61668 |
| Alternativnummer: |
TGM-T61668-1MG,TGM-T61668-5MG,TGM-T61668-10MG,TGM-T61668-25MG,TGM-T61668-50MG,TGM-T61668-100MG |
| Hersteller: |
TargetMol |
| Kategorie: |
Biochemikalien |
| GABAA receptor agent 5 demonstrates antagonist activity across multiple GABAA receptor subtypes, and GABAA receptor agent 5 exhibits IC50 values of 0.24, 0.088, 0.068, 0.33, 0.79, 0.32, 0.079, and 0.051 µM for alpha1beta2delta, alpha4beta1delta, alpha4beta2delta, alpha6beta2delta, alpha1beta2gamma2, alpha2beta2gamma2, alpha3beta2gamma2, and alpha5beta2gamma2 receptor configurations, respectively. GABAA receptor agent 5 (compound 018) thereby provides a precise pharmacological tool for characterizing subtype-selective GABAA receptor inhibition and supports mechanistic neuropharmacology studies focused on inhibitory synaptic signaling and therapeutic antagonist development. |
| Molekulargewicht: |
383.51 |
| Reinheit: |
99.39% |
| CAS Nummer: |
[1808389-92-5] |
| Formel: |
C21H25N3O2S |
| Target-Kategorie: |
GABA Receptor |
|
T61668 |
|
T61668 |