GABAA receptor agent 5, CAS [[1808389-92-5]]

Artikelnummer: TGM-T61668
Artikelname: GABAA receptor agent 5, CAS [[1808389-92-5]]
Artikelnummer: TGM-T61668
Hersteller Artikelnummer: T61668
Alternativnummer: TGM-T61668-1MG,TGM-T61668-5MG,TGM-T61668-10MG,TGM-T61668-25MG,TGM-T61668-50MG,TGM-T61668-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
GABAA receptor agent 5 demonstrates antagonist activity across multiple GABAA receptor subtypes, and GABAA receptor agent 5 exhibits IC50 values of 0.24, 0.088, 0.068, 0.33, 0.79, 0.32, 0.079, and 0.051 µM for alpha1beta2delta, alpha4beta1delta, alpha4beta2delta, alpha6beta2delta, alpha1beta2gamma2, alpha2beta2gamma2, alpha3beta2gamma2, and alpha5beta2gamma2 receptor configurations, respectively. GABAA receptor agent 5 (compound 018) thereby provides a precise pharmacological tool for characterizing subtype-selective GABAA receptor inhibition and supports mechanistic neuropharmacology studies focused on inhibitory synaptic signaling and therapeutic antagonist development.
Molekulargewicht: 383.51
Reinheit: 99.39%
CAS Nummer: [1808389-92-5]
Formel: C21H25N3O2S
Target-Kategorie: GABA Receptor
T61668
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