E6201, CAS [[603987-35-5]]
Artikelnummer:
TGM-T61755
| Artikelname: |
E6201, CAS [[603987-35-5]] |
| Artikelnummer: |
TGM-T61755 |
| Hersteller Artikelnummer: |
T61755 |
| Alternativnummer: |
TGM-T61755-25MG,TGM-T61755-50MG,TGM-T61755-100MG |
| Hersteller: |
TargetMol |
| Kategorie: |
Biochemikalien |
| E6201 (ER-806201) is a potent dual kinase inhibitor targeting MEK1 and FLT3, inhibiting their activities in an ATP-competitive manner. It effectively suppresses MEK1-induced ERK2 phosphorylation (IC50 = 5.2 nM), MKK4-induced JNK phosphorylation (IC50 = 91 nM), and MKK6-induced p38 MAPK phosphorylation (IC50 = 19 nM). E6201 exhibits anti-tumor and anti-psoriasis effects [1] [2]. |
| Molekulargewicht: |
389.44 |
| CAS Nummer: |
[603987-35-5] |
| Formel: |
C21H27NO6 |
| Target-Kategorie: |
MEK|||FLT|||Others |
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T61755 |
