TRPV1 antagonist 3 (Compound 7q) is a highly potent TRPV1 receptor antagonist with an IC50 of 2.66 nM against capsaicin. It exhibits selectivity in its mode of action, is orally bioavailable (60%), and can penetrate the central nervous system [1].
Molekulargewicht:
391.53
Formel:
C23H25N3OS
Target-Kategorie:
Others|||TRP/TRPV Channel
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