PDE4B/7A-IN-2, CAS [[2511632-55-4]]

Artikelnummer: TGM-T62064
Artikelname: PDE4B/7A-IN-2, CAS [[2511632-55-4]]
Artikelnummer: TGM-T62064
Hersteller Artikelnummer: T62064
Alternativnummer: TGM-T62064-25MG,TGM-T62064-50MG,TGM-T62064-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
This compound is a dual 5-HT1A/5-HT7 receptor antagonist (5-HT1A Ki = 8 nM, Kb = 0.04 nM, 5-HT7 Ki = 451 nM, Kb = 460 nM) with additional inhibitory activity against PDE4B/PDE7A (PDE4B IC50 = 80.4 µM, PDE7A IC50 = 151.3 µM). Its antidepressant-like effect surpasses that of the reference agent, escitalopram.
Molekulargewicht: 409.56
CAS Nummer: [2511632-55-4]
Formel: C25H35N3O2
Target-Kategorie: Others|||PDE
T62064