Prexasertib Mesylate Hydrate, CAS [[1234015-57-6]]
Artikelnummer:
TGM-T63152
| Artikelname: |
Prexasertib Mesylate Hydrate, CAS [[1234015-57-6]] |
| Artikelnummer: |
TGM-T63152 |
| Hersteller Artikelnummer: |
T63152 |
| Alternativnummer: |
TGM-T63152-25MG,TGM-T63152-50MG,TGM-T63152-100MG |
| Hersteller: |
TargetMol |
| Kategorie: |
Biochemikalien |
| Prexasertib Mesylate Hydrate (LY2606368 Mesylate Hydrate) is an ATP-competitive, selective, second-generation cell cycle checkpoint kinase 1 (CHK1) inhibitor (IC50<1 nM, Ki: 0.9 nM). It inhibits CHK2 (IC50: 8 nM) and RSK1 (IC50: 9 nM), induces double-stranded DNA breaks and replication mutations, triggers apoptosis, and exhibits potent anti-tumor effects. |
| Molekulargewicht: |
479.51 |
| CAS Nummer: |
[1234015-57-6] |
| Formel: |
C19H25N7O6S |
| Target-Kategorie: |
Apoptosis|||Chk|||Others |
|
T63152 |