Prexasertib Mesylate Hydrate, CAS [[1234015-57-6]]

Artikelnummer: TGM-T63152
Artikelname: Prexasertib Mesylate Hydrate, CAS [[1234015-57-6]]
Artikelnummer: TGM-T63152
Hersteller Artikelnummer: T63152
Alternativnummer: TGM-T63152-25MG,TGM-T63152-50MG,TGM-T63152-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
Prexasertib Mesylate Hydrate (LY2606368 Mesylate Hydrate) is an ATP-competitive, selective, second-generation cell cycle checkpoint kinase 1 (CHK1) inhibitor (IC50<1 nM, Ki: 0.9 nM). It inhibits CHK2 (IC50: 8 nM) and RSK1 (IC50: 9 nM), induces double-stranded DNA breaks and replication mutations, triggers apoptosis, and exhibits potent anti-tumor effects.
Molekulargewicht: 479.51
CAS Nummer: [1234015-57-6]
Formel: C19H25N7O6S
Target-Kategorie: Apoptosis|||Chk|||Others
T63152