CDK9-IN-19 is a selective and potent CDK9 inhibitor (IC50: 2.0 nM). CDK9-IN-19 exhibits good anti-proliferative activity in cancer cells, moderate pharmacokinetic properties and low hERG inhibition. CDK9-IN-19 significantly inhibited tumor growth in the MV4-11 xenograft mouse model. CDK9-IN-19 can be used in studies of acute myeloid leukemia (AML).
Molekulargewicht:
508.47
CAS Nummer:
[2479306-60-8]
Formel:
C26H22F2N4O5
Target-Kategorie:
CDK|||Others
T63490
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