EPI-7170 is a ralaniten analogue and a potent antagonist of the androgen receptor N-terminal structural domain, blocking the transcriptional activity of the full-length AR (FL-AR) and AR splice variants (AR-Vs). EPI-7170 exhibits antitumor activity against enzalutamide resistant debulking resistant prostate cancer (CRPC).
Molekulargewicht:
540.88
CAS Nummer:
[2139288-26-7]
Formel:
C22H28Cl3NO6S
Target-Kategorie:
Others|||Androgen Receptor
T63811
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