CDK9/10/GSK3beta-IN-1, CAS [[2423045-06-9]]

Artikelnummer: TGM-T63851
Artikelname: CDK9/10/GSK3beta-IN-1, CAS [[2423045-06-9]]
Artikelnummer: TGM-T63851
Hersteller Artikelnummer: T63851
Alternativnummer: TGM-T63851-25MG,TGM-T63851-50MG,TGM-T63851-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
CDK9/10/GSK3beta-IN-1 is a kinase inhibitor (Flavopiridol analogue) that effectively inhibits HsGSK3beta, HsCDK9/CyclinT, HsCDK5/p25 and HsCDK2/CyclinA with IC50 values of 59 nM, 64 nM, 1.093 µM and 1.725 µM, respectively. CDK9/10/GSK3beta-IN-1 exhibited comparable or higher anti-cancer cell activity than Flavopiridol and showed high anti-proliferative activity against up to seven cancer cell lines in vitro.
Molekulargewicht: 546.04
CAS Nummer: [2423045-06-9]
Formel: C29H24ClN3O4S
Target-Kategorie: Others|||CDK
T63851