I-BET282E is a pan-inhibitor of eight BET bromodomains and shows selectivity for other representative bromodomain-containing proteins. It can act on eight BRD2 (BD1/BD2), BRD2 (BD1/BD), BRD3 (BD1/BD), and BRD4 (BD1/BD), with their pIC50 values ranging from 6.4 to 7.7.
Molekulargewicht:
546.64
Formel:
C26H34N4O7S
Target-Kategorie:
Others|||Epigenetic Reader Domain
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