CYC-116, CAS [[693228-63-6]]

Artikelnummer: TGM-T6458
Artikelname: CYC-116, CAS [[693228-63-6]]
Artikelnummer: TGM-T6458
Hersteller Artikelnummer: T6458
Alternativnummer: TGM-T6458-5MG,TGM-T6458-10MG,TGM-T6458-25MG,TGM-T6458-50MG,TGM-T6458-100MG,TGM-T6458-200MG
Hersteller: TargetMol
Kategorie: Biochemikalien
CYC116 is a potent inhibitor of Aurora A/B with Ki of 8.0 nM/9.2 nM, is less potent to VEGFR2 (Ki of 44 nM), with 50-fold greater potency than CDKs, not active against PKA, Akt/PKB, PKC, no effect on GSK-3alpha/beta, CK2, Plk1 and SAPK2A. Phase 1.
Molekulargewicht: 368.46
Reinheit: 97.59%
CAS Nummer: [693228-63-6]
Formel: C18H20N6OS
Target-Kategorie: S6 Kinase|||CDK|||FLT|||Aurora Kinase|||VEGFR
T6458