EZH2-IN-15 (SHR2554) is a specific inhibitor of the zeste 2 histone modification enhancer (EZH2).EZH2 is aberrantly overexpressed in many human cancers and controls adaptive responses by regulating Treg activity. EZH2 expression in tumors has also been shown to control innate immunity.
Molekulargewicht:
548.72
Reinheit:
98.85%
CAS Nummer:
[2098545-98-1]
Formel:
C32H44N4O4
Target-Kategorie:
Histone Methyltransferase
T67883
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