OK-1035, CAS [[98293-88-0]]

Artikelnummer: TGM-T68192
Artikelname: OK-1035, CAS [[98293-88-0]]
Artikelnummer: TGM-T68192
Hersteller Artikelnummer: T68192
Alternativnummer: TGM-T68192-25MG,TGM-T68192-50MG,TGM-T68192-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
OK-1035 is a potent and selective DNA-PK inhibitor. When a synthetic peptide was used as a substrate, OK-1035 caused 50% inhibition of DNA-PK activity at 8 microM. OK-1035 inhibited the phosphorylation by DNA-PK of consensus peptide as well as that of recombinant human wild type-p53. Kinetic studies indicated that OK-1035 inhibited DNA-PK activity in an ATP-competitive manner.
Molekulargewicht: 239.23
CAS Nummer: [98293-88-0]
Formel: C12H9N5O
Target-Kategorie: Others
T68192