SKF89976A HCl, CAS [[85375-85-5]]

Artikelnummer: TGM-T68550
Artikelname: SKF89976A HCl, CAS [[85375-85-5]]
Artikelnummer: TGM-T68550
Hersteller Artikelnummer: T68550
Alternativnummer: TGM-T68550-25MG,TGM-T68550-50MG,TGM-T68550-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
SKF89976A is a potent GABA uptake inhibitor, which is selective for GAT-1 (IC50 values are 0.13, 550, 944 and 7210 µM for hGAT-1, rGAT-2, hGAT-3 and hBGT-1 respectively). SKF89976A inhibits transport current competitively (Ki = 7 µM) and transmitter-gated current non-competitively (Ki = 0.03 nM). It is able to pass the blood-brain barrier after systemic administration and is active in vivo.
Molekulargewicht: 335.44
CAS Nummer: [85375-85-5]
Formel: C22H25NO2
Target-Kategorie: Others
T68550