Encequidar, HCl, CAS [[849675-88-3]]

Produktübersicht

• Artikelname: Encequidar, HCl, CAS [[849675-88-3]]
• Artikelnummer: TGM-T68568
• Hersteller Artikelnummer: T68568
• Alternativnummer: TGM-T68568-25MG,TGM-T68568-50MG,TGM-T68568-100MG
• Hersteller: TargetMol
• Kategorie: Biochemikalien

Produktbeschreibung

Encequidar, also known as HM-30181, is an oral P-glycoprotein (P-gp) inhibitor developed to enhance the oral bioavailability of P-gp substrate drugs. Encequidar showed the highest potency (IC(50)=0.63nM) among several MDR1 inhibitors, including cycloporin A, XR9576, and GF120918, and effectively blocked transepithelial transport of paclitaxel in MDCK monolayers (IC(50)=35.4nM). Encequidar is currently under clinical trials.

Produkteigenschaften

• Molekulargewicht: 725.2
• CAS Nummer: [849675-88-3]
• Formel: C38H37ClN6O7
• Target-Kategorie: Others

Bilder

T68568