AMP423, CAS [[219501-57-2]]

Artikelnummer: TGM-T69821
Artikelname: AMP423, CAS [[219501-57-2]]
Artikelnummer: TGM-T69821
Hersteller Artikelnummer: T69821
Alternativnummer: TGM-T69821-25MG,TGM-T69821-50MG,TGM-T69821-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
AMP423 is a naphthyl derivative of 2-cyanoaziridine-1-carboxamide with structural similarity to the pro-oxidant anti-tumor agent imexon. AMP423 was active in SCID mice bearing 8226/S myeloma and SU-DHL-6 B-cell lymphoma tumors, with a median tumor growth delay (T-C) of 21 days (P = 0.0002) and 5 days (P = 0.004), respectively, and a median tumor growth inhibition (T/C) of 33.3% (P = 0.03) and 82% (P = 0.01), respectively. In non-tumor-bearing mice, AMP423 was not myelosuppressive.
Molekulargewicht: 237.26
CAS Nummer: [219501-57-2]
Formel: C14H11N3O
Target-Kategorie: Others
T69821