Milvexian TFA, CAS [[1802426-00-1]]

Artikelnummer: TGM-T70170
Artikelname: Milvexian TFA, CAS [[1802426-00-1]]
Artikelnummer: TGM-T70170
Hersteller Artikelnummer: T70170
Alternativnummer: TGM-T70170-25MG,TGM-T70170-50MG,TGM-T70170-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
Milvexian, also known as BMS-986177 and JNJ-70033093, is a blood coagulation factor XIa inhibitor. Milvexian demonstrated good selectivity over plasma kallikreinKi = 44 nM (400-fold selective), and chymotrypsinKi = 35 nM (318-fold selective). At a dose of 1.5 mg/kg, Milvexian exhibited an overall exposure of 1215 nM/h, low clearance of 10.3 mL/min/kg, and oral bioavailability of 32%.
Molekulargewicht: 742.49
CAS Nummer: [1802426-00-1]
Formel: C30H26Cl2F5N9O4
Target-Kategorie: Others|||Factor Xa
T70170