PF-04479745, also known as PF-4479745, is a potent and selective 5-HT2C agonist (EC50 = 10 nM). PF-4479745 displayed robust pharmacology in a preclinical canine model of stress urinary incontinence (SUI) and no measurable functional agonism at the key selectivity targets 5-HT2A and 5-HT2B in relevant tissue-based assay systems.
Molekulargewicht:
432.477
CAS Nummer:
[1613691-76-1]
Formel:
C21H28N4O6
Target-Kategorie:
Others
T70379
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