ML252 is a selective potassium channel inhibitor, specifically targeting the KCNQ2 channel (Kv7.2) with an IC50 value of 69 nM. Additionally, ML252 demonstrates inhibitory activity against Cytochrome P450 isoforms, including IC50 values of 6.1 nM (CYP1A2), 18.9 nM (CYP2C9), 3.9 nM (CYP3A4), and 19.9 nM (CYP2D6).
Molekulargewicht:
308.42
CAS Nummer:
[1392494-64-2]
Formel:
C20H24N2O
Target-Kategorie:
Cytochromes P450|||Potassium Channel|||Others
T70786
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