Rimegepant, also known as BMS-927711 and BHV-3000, is a potent, selective, competitive, and orally active calcitonin gene-related peptide (CGRP) antagonist in clinical trials for treating migraines. Rimegepant has shown in vivo efficacy without vasoconstriction effect. BMS-927711 is superior to placebo at several different doses (75 mg, 150 mg, and 300 mg) and has an excellent tolerability profile.
Molekulargewicht:
1221.2526
CAS Nummer:
[1374024-48-2]
Formel:
C56H64F4N12O13S
Target-Kategorie:
Others|||CGRP Receptor
T70837
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