Syntelin, CAS [[438481-33-5]]

Artikelnummer: TGM-T71828
Artikelname: Syntelin, CAS [[438481-33-5]]
Artikelnummer: TGM-T71828
Hersteller Artikelnummer: T71828
Alternativnummer: TGM-T71828-25MG,TGM-T71828-50MG,TGM-T71828-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
Syntelin is a selectively CENP-E inhibitor. Syntelin inhibited CENP-E motility in a dose-dependent manner with an IC50 value of 160 nM. Among an extensive list of mitotic kinesins examined, syntelin was found to be highly selective for CENP-E. Syntelin binds to different sites from those of GSK923295, a recently identified CENP-E ATPase inhibitor, as syntelin inhibits CENP-E mutants resistant to GSK923295 in a manner indistinguishable from that of wild type motor. Syntelin represents a novel class of CENP-E motor inhibitor.
Molekulargewicht: 484.62
CAS Nummer: [438481-33-5]
Formel: C21H20N6O2S3
Target-Kategorie: Others|||Kinesin
T71828