beta2AR/M-receptor agonist-2, CAS [[1017857-38-3]]
Artikelnummer:
TGM-T72226
Hersteller Artikelnummer:
T72226
Alternativnummer:
TGM-T72226-25MG,TGM-T72226-50MG,TGM-T72226-100MG
Hersteller:
TargetMol
Kategorie:
Biochemikalien
beta2AR/M-receptor agonist-2 is a dual-function compound acting as a muscarinic antagonist and beta2 adrenoceptor agonist (MABA). It demonstrates significant activity towards the beta2 adrenoceptor with an EC50 of 3.7 nM and exhibits affinity for the human cloned M3 receptor with a Ki of 0.73 nM. This potent bronchodilator holds potential for research in chronic obstructive pulmonary disease (COPD) treatment.
Molekulargewicht:
717.31
CAS Nummer:
[1017857-38-3]
Formel:
C36H49ClN4O7S
Target-Kategorie:
AChR|||Others|||Adrenergic Receptor
T72226
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