EZH2-IN-14 is a selective inhibitor of EZH2 (Histone Methyltransferase) with an IC50 value of 12 nM, targeting the methyltransferase activity of EZH2/PRC2 and reducing H3K27me3 levels. It exhibits more than 200-fold selectivity for EZH2 over the closely related H3K27 methyltransferase, EZH1.
Molekulargewicht:
541.69
CAS Nummer:
[1979157-17-9]
Formel:
C31H39N7O2
Target-Kategorie:
Histone Methyltransferase|||Others
T73134
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