MRS4719, CAS [[2840581-32-8]]

Artikelnummer: TGM-T73453
Artikelname: MRS4719, CAS [[2840581-32-8]]
Artikelnummer: TGM-T73453
Hersteller Artikelnummer: T73453
Alternativnummer: TGM-T73453-25MG,TGM-T73453-50MG,TGM-T73453-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
MRS4719, a potent P2X4 receptor antagonist, exhibits a half-maximal inhibitory concentration (IC50) of 0.503 µM for the human P2X4 receptor. Demonstrating both neuroprotective and neuro-rehabilitative effects, it can decrease infarct volume and brain atrophy in an ischemic stroke model. Additionally, MRS4719 mitigates ATP-induced calcium influx in primary human monocyte-derived macrophages, making it a valuable tool for researching ischemic stroke.
Molekulargewicht: 504.6
CAS Nummer: [2840581-32-8]
Formel: C26H13N5O3S.C6H15N
Target-Kategorie: Others|||P2X Receptor
T73453