AZ6421, functioning as a Proteolysis Targeting Chimera (PROTAC), selectively degrades estrogen receptor alpha, demonstrating potent anti-tumor activity by inhibiting uncontrolled cellular proliferation characteristic of malignant diseases. This compound holds promise for cancer research, including breast cancer applications [1].
Molekulargewicht:
975.17
CAS Nummer:
[2361115-35-5]
Formel:
C52H65F3N6O7S
Target-Kategorie:
Estrogen Receptor/ERR|||PROTACs|||Others
T74060
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