PROTAC EZH2 Degrader-1, CAS [[2641601-67-2]]

Artikelnummer: TGM-T74602
Artikelname: PROTAC EZH2 Degrader-1, CAS [[2641601-67-2]]
Artikelnummer: TGM-T74602
Hersteller Artikelnummer: T74602
Alternativnummer: TGM-T74602-1MG,TGM-T74602-5MG,TGM-T74602-10MG
Hersteller: TargetMol
Kategorie: Biochemikalien
PROTAC EZH2 Degrader-1 (Compound 150d) is a potent PROTAC molecule that effectively suppresses EZH2 methyltransferase activity, with a half-maximal IC50 of 2.7 nM. EZH2 is a histone methyltransferase crucial to tumorigenesis and cancer progression, and PROTAC EZH2 Degrader-1 represents an important chemical tool for probing its therapeutic relevance.
Molekulargewicht: 942.15
CAS Nummer: [2641601-67-2]
Formel: C54H67N7O8
Target-Kategorie: PROTACs|||Histone Methyltransferase
T74602
T74602