PROTAC EZH2 Degrader-1 (Compound 150d) is a potent PROTAC molecule that effectively suppresses EZH2 methyltransferase activity, with a half-maximal IC50 of 2.7 nM. EZH2 is a histone methyltransferase crucial to tumorigenesis and cancer progression, and PROTAC EZH2 Degrader-1 represents an important chemical tool for probing its therapeutic relevance.
Molekulargewicht:
942.15
CAS Nummer:
[2641601-67-2]
Formel:
C54H67N7O8
Target-Kategorie:
PROTACs|||Histone Methyltransferase
T74602
T74602
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