NC-III-49-1, CAS [[3031654-46-0]]

Artikelnummer: TGM-T74898
Artikelname: NC-III-49-1, CAS [[3031654-46-0]]
Artikelnummer: TGM-T74898
Hersteller Artikelnummer: T74898
Alternativnummer: TGM-T74898-1MG,TGM-T74898-5MG,TGM-T74898-10MG,TGM-T74898-25MG,TGM-T74898-50MG,TGM-T74898-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
NC-III-49-1 is a potent bivalent bromodomain and extraterminal domain (BET) inhibitor with significant affinity for various BRD4 and BRDT isoforms, as demonstrated by its Kd values of 0.095 nM for BRD4-1, 0.32 nM for BRD4-2, 0.29 nM for BRD4-T, 0.089 nM for BRDT-1, 5.5 nM for BRDT-2, and 0.058 nM for BRDT-T. Additionally, NC-III-49-1 exhibits antiproliferative effects and reduces the expression of c-Myc [1].
Molekulargewicht: 875.02
CAS Nummer: [3031654-46-0]
Formel: C44H50N4O11S2
Target-Kategorie: Others|||Epigenetic Reader Domain
T74898