ELA-11(human) TFA, a bioactive fragment of ELA-32, acts as a high-affinity apelin receptor agonist (K i =14 nM). It effectively inhibits forskolin-induced cAMP production and promotes beta-arrestin recruitment in vitro, highlighting its significant agonistic activity.
Molekulargewicht:
1397.58
Formel:
C60H91F3N16O15S2
Target-Kategorie:
Apelin receptor
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