(E/Z)-GSK5182, CAS [[2699724-40-6]]
Artikelnummer:
TGM-T7709
- Bilder (1)
| Artikelname: | (E/Z)-GSK5182, CAS [[2699724-40-6]] |
| Artikelnummer: | TGM-T7709 |
| Hersteller Artikelnummer: | T7709 |
| Alternativnummer: | TGM-T7709-1MLX10MM(INDMSO),TGM-T7709-1MG,TGM-T7709-5MG,TGM-T7709-10MG,TGM-T7709-25MG,TGM-T7709-50MG,TGM-T7709-100MG |
| Hersteller: | TargetMol |
| Kategorie: | Biochemikalien |
| Alternative Synonym: | GSK5182(Z/E) |
| (E/Z)-GSK5182 (GSK5182(Z/E)) is a racemic mixture comprising (E)-GSK5182 and (Z)-GSK5182 isomers. It acts as a highly selective and orally active inverse agonist for the estrogen-related receptor gamma (ERRgamma), demonstrating potency with an IC50 of 79 nM. Additionally, GSK5182 is known to induce the generation of reactive oxygen species (ROS) in hepatocellular carcinoma. |
| Molekulargewicht: | 417.54 |
| Reinheit: | 97.58% |
| CAS Nummer: | [2699724-40-6] |
| Formel: | C27H31NO3 |
| Target-Kategorie: | Estrogen Receptor/ERR|||Estrogen/progestogen Receptor|||Reactive Oxygen Species|||ROS |

