A-77636 is a potent, selective, and long-acting oral dopamine D1 receptor agonist with an effective concentration (EC50) of 1.1 nM and a corresponding pEC50 value of 8.13. It demonstrates the highest affinity for the dopamine D1 receptor with a dissociation constant (Ki) of 39.8 nM and a pKi of 7.40 0.09. Notably, A-77636 exhibits antiparkinsonian activity [1].
Molekulargewicht:
329.43
CAS Nummer:
[778546-51-3]
Formel:
C20H27NO3
Target-Kategorie:
Dopamine Receptor
T78644
* Mehrwertsteuer und Versandkosten nicht enthalten. Irrtümer und Preisänderungen vorbehalten
