FGFR-IN-11, CAS [[2658488-68-5]]

Artikelnummer: TGM-T79257
Artikelname: FGFR-IN-11, CAS [[2658488-68-5]]
Artikelnummer: TGM-T79257
Hersteller Artikelnummer: T79257
Alternativnummer: TGM-T79257-25MG,TGM-T79257-50MG,TGM-T79257-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
FGFR-IN-11 (compound I-5) is an orally active, covalent inhibitor of FGFR, with IC50 values of 9.9 nM (FGFR1), 3.1 nM (FGFR2), 16 nM (FGFR3), and 1.8 nM (FGFR4). This compound demonstrates nanomolar potency in inhibiting the proliferation of various cancer cells and significantly hinders tumor growth in xenograft mouse models [1].
Molekulargewicht: 521.01
CAS Nummer: [2658488-68-5]
Formel: C28H29ClN4O4
Target-Kategorie: FGFR
T79257