ER degrader 7, CAS [[2922929-63-1]] Preis auf Anfrage
Artikelnummer:
TGM-T79383
Hersteller Artikelnummer:
T79383
Alternativnummer:
TGM-T79383-5MG,TGM-T79383-50MG
Hersteller:
TargetMol
Kategorie:
Biochemikalien
ER degrader 7 (Compound 35t) is a selective degrader of both ERalpha and ERbeta and functions as a tubulin polymerization inhibitor. It inhibits cell viability with IC50 values of 0.06 µM for MCF-7, 2.56 µM for T47D, 15.84 µM for MCF-10A, 1.59 µM for LCC2, 1.67 µM for T47D D538G, and 1.37 µM for T47D Y537S cells. Additionally, ER degrader 7 demonstrates efficacy in suppressing breast cancer tumor growth [1].