Rezatapopt (PC14586) is a small molecule p53 reactivator with anti-tumor activity that selectively binds to the cleft present in the TP53 Y220C mutant protein and restores the p53 wild-type (normal) conformation and transcriptional activity, and can be used to study locally advanced or metastatic solid tumors.
Molekulargewicht:
545.57
Reinheit:
98.12%
CAS Nummer:
[2636846-41-6]
Formel:
C28H31F4N5O2
Target-Kategorie:
Others|||MDM-2/p53|||p53
T81289
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