Pomalidomide-C5-Dovitinib, CAS [[2732969-67-2]] Preis auf Anfrage
Artikelnummer:
TGM-T81421
Hersteller Artikelnummer:
T81421
Alternativnummer:
TGM-T81421-5MG,TGM-T81421-50MG
Hersteller:
TargetMol
Kategorie:
Biochemikalien
Pomalidomide-C5-Dovitinib (compound 2) is a PROTAC linking Pomalidomide and Dovitinib via a CRBN connector, exhibiting potent antiproliferative activity in FLT3-ITD+ acute myeloid leukemia (AML) cells. It promotes ubiquitin-proteasome-dependent degradation of FLT3-ITD and KIT proteins, thereby inhibiting their downstream signaling pathways and presenting research potential in FLT3-ITD+ AML [1].