KSL-128114 TFA

Artikelnummer: TGM-T83716
Artikelname: KSL-128114 TFA
Artikelnummer: TGM-T83716
Hersteller Artikelnummer: T83716
Alternativnummer: TGM-T83716-1MG,TGM-T83716-5MG,TGM-T83716-10MG,TGM-T83716-25MG
Hersteller: TargetMol
Kategorie: Biochemikalien
Alternative Synonym: Ac-rRrGrKkRrSHWX1X2DI-OH (X1=tert-Leucine, X2=Cyclohexylglycine)
KSL-128114, a peptide inhibitor of the membrane regulator syntenin (Ki = 300 nM), notably diminishes the viability of A2058 melanoma and patient-derived glioblastoma multiforme (GBM) cells in a concentration-dependent manner. Furthermore, when administered at 50 µM, KSL-128114 elevates survival times in a patient-derived xenograft (PDX) mouse model of GBM, where mice were implanted intracranially with patient-derived GBM cells pre-cultured with KSL-128114.
Molekulargewicht: 2201.6
Formel: C96H165N39O21.XCF3COOH
T83716