BPR5K230, CAS [[3029897-97-7]]

Artikelnummer: TGM-T88671
Artikelname: BPR5K230, CAS [[3029897-97-7]]
Artikelnummer: TGM-T88671
Hersteller Artikelnummer: T88671
Alternativnummer: TGM-T88671-25MG,TGM-T88671-50MG,TGM-T88671-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
BPR5K230 is a dual inhibitor of the receptor tyrosine kinases MER and AXL, exhibiting IC50 values of 4.1 nM and 9.2 nM, respectively. It inhibits the proliferation of Ba/F3-MER cells with an IC50 of 5 nM. BPR5K230 demonstrates favorable pharmacokinetics in mice and displays anti-inflammatory and antitumor effects in mouse models against 4T1, MDA-MB-231, MC38, and Hepa1-6.
Molekulargewicht: 655.68
CAS Nummer: [3029897-97-7]
Formel: C37H30FN7O4
Target-Kategorie: TAM Receptor
T88671