Transcription factor-IN-1 (Compound 4e) acts as an inhibitor of transcription factors. It exhibits anticonvulsant activity by antagonizing pentylenetetrazole (PTZ) with an ED50 of 34.5 mg/kg. Additionally, Transcription factor-IN-1 demonstrates antidepressant activity in a rat model.
Target-Kategorie:
GABA Receptor|||Others
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