IRE1alpha kinase-IN-1, CAS [[2328097-41-0]]

Artikelnummer: TGM-T9564
Artikelname: IRE1alpha kinase-IN-1, CAS [[2328097-41-0]]
Artikelnummer: TGM-T9564
Hersteller Artikelnummer: T9564
Alternativnummer: TGM-T9564-1MLX10MM(INDMSO),TGM-T9564-1MG,TGM-T9564-5MG,TGM-T9564-10MG,TGM-T9564-25MG,TGM-T9564-50MG,TGM-T9564-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
IRE1alpha kinase-IN-1 is a highly selective IRE1alpha (ERN1) inhibitor, with an IC50 of 77 nM, displaying 100-fold selectivity over the IRE1beta isoform. It inhibits ER stress-induced IRE1alpha oligomerization and autophosphorylation, as well as IRE1alpha RNase activity (IC50=80 nM).
Molekulargewicht: 504.99
Reinheit: 99.18%
CAS Nummer: [2328097-41-0]
Formel: C26H26ClFN8
Target-Kategorie: IRE1
T9564