IRE1alpha kinase-IN-1, CAS [[2328097-41-0]]
Artikelnummer:
TGM-T9564
- Bilder (1)
| Artikelname: | IRE1alpha kinase-IN-1, CAS [[2328097-41-0]] |
| Artikelnummer: | TGM-T9564 |
| Hersteller Artikelnummer: | T9564 |
| Alternativnummer: | TGM-T9564-1MLX10MM(INDMSO),TGM-T9564-1MG,TGM-T9564-5MG,TGM-T9564-10MG,TGM-T9564-25MG,TGM-T9564-50MG,TGM-T9564-100MG |
| Hersteller: | TargetMol |
| Kategorie: | Biochemikalien |
| IRE1alpha kinase-IN-1 is a highly selective IRE1alpha (ERN1) inhibitor, with an IC50 of 77 nM, displaying 100-fold selectivity over the IRE1beta isoform. It inhibits ER stress-induced IRE1alpha oligomerization and autophosphorylation, as well as IRE1alpha RNase activity (IC50=80 nM). |
| Molekulargewicht: | 504.99 |
| Reinheit: | 99.18% |
| CAS Nummer: | [2328097-41-0] |
| Formel: | C26H26ClFN8 |
| Target-Kategorie: | IRE1 |

