[Des-His1,Glu9]-Glucagon amide, CAS [[110084-95-2]]
Artikelnummer:
TGM-TP2033
Hersteller Artikelnummer:
TP2033
Alternativnummer:
TGM-TP2033-1MG
Hersteller:
TargetMol
Kategorie:
Biochemikalien
Alternative Synonym:
des-His1-[Glu9]-Glucagon (1-29) amide
Glucagon receptor antagonist (pA2 = 7.2 for inhibition of glucagon-induced adenylyl cyclase activation in rat liver membranes), displays no agonist activity. Enhances glucose-stimulated pancreatic insulin release in vitro. Blocks added glucagon-induced hyperglycemia in normal rabbits without affecting glycogenolysis in vivo. Also blocks endogenous glucagon-induced hyperglycemia in streptozocin diabetic rats.
Molekulargewicht:
3358.68
CAS Nummer:
[110084-95-2]
Formel:
C148H221N41O47S
Target-Kategorie:
Glucagon Receptor
TP2033
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