Urotensin-II (UT) receptor ligand, behaves as a silent antagonist in most in vitro assays and in vivo, but does retain small residual agonist activity under certain conditions in some assays. Competitively antagonizes U-II induced contractions in the rat aorta (pIC50 = 7.46) and prevents plasma extravasation elicited by U-II in mice in vivo.
Molekulargewicht:
1061.24
CAS Nummer:
[879497-82-2]
Formel:
C50H64N10O12S2
Target-Kategorie:
GPCR
TP2104
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